Discovery and early optimization of 1H-indole-2-carboxamides with anti-trypanosoma cruzi activity (2025)
- Authors:
- USP affiliated authors: DUARTE, SIMONE MICHELAN - IFSC ; ANDRICOPULO, RENATA KROGH - IFSC ; FERREIRA, LEONARDO LUIZ GOMES - IFSC ; FREITAS, CAROLINA BORSOI MORAES HOLANDA DE - FCF ; ANDRICOPULO, ADRIANO DEFINI - IFSC ; CHELUCCI, RAFAEL CONSOLIN - IFSC ; FELTRIN, CLARISSA - ICB ; SILVA, ADRIANA CORRÊA DA - ICB ; SANTOS, BENEDITO MATHEUS DOS - FCF ; BROERING, MILENA FRONZA - FCF
- Unidades: IFSC; FCF; ICB
- DOI: 10.1021/acs.jmedchem.4c02942
- Subjects: DOENÇA DE CHAGAS; QUÍMICA MÉDICA; PLANEJAMENTO DE FÁRMACOS; ANTIPARASITÁRIOS; TRYPANOSOMA CRUZI
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Publisher place: Washington, DC
- Date published: 2025
- Source:
- Título: Journal of Medicinal Chemistry
- ISSN: 0022-2623
- Volume/Número/Paginação/Ano: v. 68, n. 7, p. 7313-7340 + supporting information, Apr. 2025
- Este periódico é de assinatura
- Este artigo é de acesso aberto
- URL de acesso aberto
- Cor do Acesso Aberto: hybrid
- Licença: cc-by
-
ABNT
OLIVEIRA, Ramon Guerra de et al. Discovery and early optimization of 1H-indole-2-carboxamides with anti-trypanosoma cruzi activity. Journal of Medicinal Chemistry, v. 68, n. 7, p. 7313-7340 + supporting information, 2025Tradução . . Disponível em: https://doi.org/10.1021/acs.jmedchem.4c02942. Acesso em: 29 dez. 2025. -
APA
Oliveira, R. G. de, Duarte, S. M., Krogh, R., Ferreira, L. L. G., Chelucci, R. C., Feltrin, C., et al. (2025). Discovery and early optimization of 1H-indole-2-carboxamides with anti-trypanosoma cruzi activity. Journal of Medicinal Chemistry, 68( 7), 7313-7340 + supporting information. doi:10.1021/acs.jmedchem.4c02942 -
NLM
Oliveira RG de, Duarte SM, Krogh R, Ferreira LLG, Chelucci RC, Feltrin C, Silva AC da, Santos BM dos, Broering MF, Moraes CB, Andricopulo AD. Discovery and early optimization of 1H-indole-2-carboxamides with anti-trypanosoma cruzi activity [Internet]. Journal of Medicinal Chemistry. 2025 ; 68( 7): 7313-7340 + supporting information.[citado 2025 dez. 29 ] Available from: https://doi.org/10.1021/acs.jmedchem.4c02942 -
Vancouver
Oliveira RG de, Duarte SM, Krogh R, Ferreira LLG, Chelucci RC, Feltrin C, Silva AC da, Santos BM dos, Broering MF, Moraes CB, Andricopulo AD. Discovery and early optimization of 1H-indole-2-carboxamides with anti-trypanosoma cruzi activity [Internet]. Journal of Medicinal Chemistry. 2025 ; 68( 7): 7313-7340 + supporting information.[citado 2025 dez. 29 ] Available from: https://doi.org/10.1021/acs.jmedchem.4c02942 - Antitrypanosomal Benzoxazinone series: hit-to-lead campaign and multiparametric optimization
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Informações sobre o DOI: 10.1021/acs.jmedchem.4c02942 (Fonte: oaDOI API)
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