Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum (2024)
- Authors:
- Lapierre, Thibault Joseph William Jacques Dit
- Farago, Danilo Nascimento
- Cruz, Mariza Gabriela Faleiro de Moura Lodi
- Resende, Daniela de Melo
- Oliveira, Adriane Cristina Rosa de
- Santos, Brenda Rosa Macedo dos
- Souza, Felipe de Oliveira
- Duarte, Simone Michelan
- Chelucci, Rafael Consolin
- Andricopulo, Adriano Defini
- Ferreira, Leonardo Luiz Gomes
- Pilau, Eduardo Jorge
- Murta, Silvane M. F.
- Rezende Junior, Celso de Oliveira
- Lapierre, Thibault Joseph William Jacques Dit
- USP affiliated authors: DUARTE, SIMONE MICHELAN - IFSC ; ANDRICOPULO, ADRIANO DEFINI - IFSC ; FERREIRA, LEONARDO LUIZ GOMES - IFSC ; CHELUCCI, RAFAEL CONSOLIN - IFSC
- Unidade: IFSC
- DOI: 10.1111/cbdd.14525
- Subjects: LEISHMANIA; MECANISMOS DE DEFESA; TRYPANOSOMA CRUZI
- Keywords: ADME; Benzothiazoles; SelA; Hit discovery; Leishmania infantum
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Source:
- Título: Chemical Biology and Drug Design
- ISSN: 1747-0285
- Volume/Número/Paginação/Ano: v. 103, p. e14525-1-e14525-14 + supporting information, Apr. 2024
- Este periódico é de acesso aberto
- Este artigo NÃO é de acesso aberto
-
ABNT
LAPIERRE, Thibault Joseph William Jacques Dit et al. Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum. Chemical Biology and Drug Design, v. 103, p. e14525-1-e14525-14 + supporting information, 2024Tradução . . Disponível em: https://doi.org/10.1111/cbdd.14525. Acesso em: 10 fev. 2026. -
APA
Lapierre, T. J. W. J. D., Farago, D. N., Cruz, M. G. F. de M. L., Resende, D. de M., Oliveira, A. C. R. de, Santos, B. R. M. dos, et al. (2024). Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum. Chemical Biology and Drug Design, 103, e14525-1-e14525-14 + supporting information. doi:10.1111/cbdd.14525 -
NLM
Lapierre TJWJD, Farago DN, Cruz MGF de ML, Resende D de M, Oliveira ACR de, Santos BRM dos, Souza F de O, Duarte SM, Chelucci RC, Andricopulo AD, Ferreira LLG, Pilau EJ, Murta SMF, Rezende Junior C de O. Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum [Internet]. Chemical Biology and Drug Design. 2024 ; 103 e14525-1-e14525-14 + supporting information.[citado 2026 fev. 10 ] Available from: https://doi.org/10.1111/cbdd.14525 -
Vancouver
Lapierre TJWJD, Farago DN, Cruz MGF de ML, Resende D de M, Oliveira ACR de, Santos BRM dos, Souza F de O, Duarte SM, Chelucci RC, Andricopulo AD, Ferreira LLG, Pilau EJ, Murta SMF, Rezende Junior C de O. Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum [Internet]. Chemical Biology and Drug Design. 2024 ; 103 e14525-1-e14525-14 + supporting information.[citado 2026 fev. 10 ] Available from: https://doi.org/10.1111/cbdd.14525 - Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas disease
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Informações sobre o DOI: 10.1111/cbdd.14525 (Fonte: oaDOI API)
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