Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium (2022)
- Authors:
- Cruz, Luiza
- Silva, Adriana Corrêa da
- Feltrin, Clarissa
- Dichiara, Maria
- Ferrins, Lori
- Moraes, Carolina Borsoi
- Sjo, Peter
- Andricopulo, Adriano Defini
- Mowbray, Charles
- Oliveira, Ramon Guerra de
- Dessoy, Marco Aurélio
- Santos, Deborah Araújo dos
- Oliveira, Luiz Fernando Nascimento de
- Mollo, María Cruz
- Lee, Eun
- Duarte, Simone Michelan
- Krogh, Renata
- Chelucci, Rafael Consolin
- Ferreira, Leonardo Luiz Gomes
- Kratz, Jadel Muller
- Dias, Luiz Carlos
- USP affiliated authors: ANDRICOPULO, ADRIANO DEFINI - IFSC ; DUARTE, SIMONE MICHELAN - IFSC ; ANDRICOPULO, RENATA KROGH - IFSC ; CHELUCCI, RAFAEL CONSOLIN - IFSC ; FERREIRA, LEONARDO LUIZ GOMES - IFSC
- Unidade: IFSC
- Subjects: DOENÇAS NEGLIGENCIADAS; DOENÇA DE CHAGAS
- Keywords: Phenotypic screening; Drug Discovery; Medicinal Chemistry; Indoles; CYP51 inhibition
- Language: Inglês
- Imprenta:
- Source:
- Título: Anais eletrônicos
- Conference titles: Brazilian Symposium on Medicinal Chemistry - BrazMedChem
-
ABNT
CRUZ, Luiza et al. Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium. 2022, Anais.. Campinas: Galoá, 2022. Disponível em: https://proceedings.science/brazmedchem-2022/papers/indoles-hit-to-lead-for-chagas-disease---lessons-learned-within-the-lola-consortium. Acesso em: 31 mar. 2026. -
APA
Cruz, L., Silva, A. C. da, Feltrin, C., Dichiara, M., Ferrins, L., Moraes, C. B., et al. (2022). Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium. In Anais eletrônicos. Campinas: Galoá. Recuperado de https://proceedings.science/brazmedchem-2022/papers/indoles-hit-to-lead-for-chagas-disease---lessons-learned-within-the-lola-consortium. -
NLM
Cruz L, Silva AC da, Feltrin C, Dichiara M, Ferrins L, Moraes CB, Sjo P, Andricopulo AD, Mowbray C, Oliveira RG de, Dessoy MA, Santos DA dos, Oliveira LFN de, Mollo MC, Lee E, Duarte SM, Krogh R, Chelucci RC, Ferreira LLG, Kratz JM, Dias LC. Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium [Internet]. Anais eletrônicos. 2022 ;[citado 2026 mar. 31 ] Available from: https://proceedings.science/brazmedchem-2022/papers/indoles-hit-to-lead-for-chagas-disease---lessons-learned-within-the-lola-consortium. -
Vancouver
Cruz L, Silva AC da, Feltrin C, Dichiara M, Ferrins L, Moraes CB, Sjo P, Andricopulo AD, Mowbray C, Oliveira RG de, Dessoy MA, Santos DA dos, Oliveira LFN de, Mollo MC, Lee E, Duarte SM, Krogh R, Chelucci RC, Ferreira LLG, Kratz JM, Dias LC. Indoles hit-to-lead for chagas disease: lessons learned within the LOLA consortium [Internet]. Anais eletrônicos. 2022 ;[citado 2026 mar. 31 ] Available from: https://proceedings.science/brazmedchem-2022/papers/indoles-hit-to-lead-for-chagas-disease---lessons-learned-within-the-lola-consortium. - Convergent synthesis of proline-functionalized pyrazolopyrimidines as anti-T. cruzi bioactive compounds
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