Antitrypanosomal Benzoxazinone series: hit-to-lead campaign and multiparametric optimization (2022)
- Authors:
- Mollo, María Cruz
- Cruz, Luiza
- Dessoy, Marco Aurélio
- Lee, Eun
- Oliveira, Ramon Guerra de
- Dutra, Francielle
- Duarte, Simone Michelan
- Andricopulo, Renata Krogh
- Ferreira, Leonardo Luiz Gomes
- Chelucci, Rafael Consolin
- Feltrin, Clarissa
- Moraes, Carolina Borsoi
- Andricopulo, Adriano Defini
- Kratz, Jadel
- Sjö, Peter
- Mowbray, Charles
- Dias, Luiz Carlos
- USP affiliated authors: ANDRICOPULO, ADRIANO DEFINI - IFSC ; ANDRICOPULO, RENATA KROGH - IFSC ; DUARTE, SIMONE MICHELAN - IFSC ; FERREIRA, LEONARDO LUIZ GOMES - IFSC ; CHELUCCI, RAFAEL CONSOLIN - IFSC ; FELTRIN, CLARISSA - ICB
- Unidades: IFSC; ICB
- Subjects: TRYPANOSOMA CRUZI; PLANEJAMENTO DE FÁRMACOS
- Keywords: Chagas disease; Benzoxazinones; Drug Discovery; SAR; Phenotypic screening
- Language: Inglês
- Imprenta:
- Source:
- Título: Anais eletrônicos
- Conference titles: Brazilian Symposium on Medicinal Chemistry - BrazMedChem
-
ABNT
MOLLO, María Cruz et al. Antitrypanosomal Benzoxazinone series: hit-to-lead campaign and multiparametric optimization. 2022, Anais.. Campinas: Galoá, 2022. Disponível em: https://proceedings.science/brazmedchem-2022/papers/antitrypanosomal-benzoxazinone-series--hit-to-lead-campaign-and-multiparametric-optimization-. Acesso em: 27 dez. 2025. -
APA
Mollo, M. C., Cruz, L., Dessoy, M. A., Lee, E., Oliveira, R. G. de, Dutra, F., et al. (2022). Antitrypanosomal Benzoxazinone series: hit-to-lead campaign and multiparametric optimization. In Anais eletrônicos. Campinas: Galoá. Recuperado de https://proceedings.science/brazmedchem-2022/papers/antitrypanosomal-benzoxazinone-series--hit-to-lead-campaign-and-multiparametric-optimization-. -
NLM
Mollo MC, Cruz L, Dessoy MA, Lee E, Oliveira RG de, Dutra F, Duarte SM, Andricopulo RK, Ferreira LLG, Chelucci RC, Feltrin C, Moraes CB, Andricopulo AD, Kratz J, Sjö P, Mowbray C, Dias LC. Antitrypanosomal Benzoxazinone series: hit-to-lead campaign and multiparametric optimization [Internet]. Anais eletrônicos. 2022 ;[citado 2025 dez. 27 ] Available from: https://proceedings.science/brazmedchem-2022/papers/antitrypanosomal-benzoxazinone-series--hit-to-lead-campaign-and-multiparametric-optimization-. -
Vancouver
Mollo MC, Cruz L, Dessoy MA, Lee E, Oliveira RG de, Dutra F, Duarte SM, Andricopulo RK, Ferreira LLG, Chelucci RC, Feltrin C, Moraes CB, Andricopulo AD, Kratz J, Sjö P, Mowbray C, Dias LC. Antitrypanosomal Benzoxazinone series: hit-to-lead campaign and multiparametric optimization [Internet]. Anais eletrônicos. 2022 ;[citado 2025 dez. 27 ] Available from: https://proceedings.science/brazmedchem-2022/papers/antitrypanosomal-benzoxazinone-series--hit-to-lead-campaign-and-multiparametric-optimization-. - Convergent synthesis of proline-functionalized pyrazolopyrimidines as anti-T. cruzi bioactive compounds
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