ReP USP - Resultado da busca

Trabalho de evento-resumo
Design, synthesis and in vitro evaluation of a series of arylmorpholine derivative compounds against chagas disease (2025)
Farago, Danilo Nascimento; Resende, Daniela de Melo ; Chelucci, Rafael Consolin ; Andricopulo, Adriano Defini ; Ferreira, Leonardo Luiz Gomes ; Murta, Silvane Maria Fonseca ; Rezende Junior, Celso de Oliveira
Source: Anais. Conference titles: Reunião Anual da Sociedade Brasileira de Química - RASBQ. Unidade: IFSC
Subjects: PLANEJAMENTO DE FÁRMACOS, DOENÇA DE CHAGAS
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ABNT
FARAGO, Danilo Nascimento et al. Design, synthesis and in vitro evaluation of a series of arylmorpholine derivative compounds against chagas disease. 2025, Anais.. São Paulo: Sociedade Brasileira de Química - SBQ, 2025. Disponível em: https://repositorio.usp.br/directbitstream/488b6113-cf75-4d55-a443-c3d253019b10/3259726.pdf. Acesso em: 08 out. 2025.
APA
Farago, D. N., Resende, D. de M., Chelucci, R. C., Andricopulo, A. D., Ferreira, L. L. G., Murta, S. M. F., & Rezende Junior, C. de O. (2025). Design, synthesis and in vitro evaluation of a series of arylmorpholine derivative compounds against chagas disease. In Anais. São Paulo: Sociedade Brasileira de Química - SBQ. Recuperado de https://repositorio.usp.br/directbitstream/488b6113-cf75-4d55-a443-c3d253019b10/3259726.pdf
NLM
Farago DN, Resende D de M, Chelucci RC, Andricopulo AD, Ferreira LLG, Murta SMF, Rezende Junior C de O. Design, synthesis and in vitro evaluation of a series of arylmorpholine derivative compounds against chagas disease [Internet]. Anais. 2025 ;[citado 2025 out. 08 ] Available from: https://repositorio.usp.br/directbitstream/488b6113-cf75-4d55-a443-c3d253019b10/3259726.pdf
Vancouver
Farago DN, Resende D de M, Chelucci RC, Andricopulo AD, Ferreira LLG, Murta SMF, Rezende Junior C de O. Design, synthesis and in vitro evaluation of a series of arylmorpholine derivative compounds against chagas disease [Internet]. Anais. 2025 ;[citado 2025 out. 08 ] Available from: https://repositorio.usp.br/directbitstream/488b6113-cf75-4d55-a443-c3d253019b10/3259726.pdf
Trabalho de evento-resumo
Hit-to-Lead optimization of pyridylpiperazine derivatives: promising antimalarial candidates with notable ADME profiles and metabolic stability (2025)
Oliveira, Douglas Davison da Silva ; Krüger, Arne ; Chelucci, Rafael Consolin ; Ferreira, Leonardo Luiz Gomes ; Andricopulo, Adriano Defini ; Wunderlich, Gerhard ; Silva, Neide Maria da; Rezende Junior, Celso de Oliveira
Source: Anais. Conference titles: Reunião Anual da Sociedade Brasileira de Química - RASBQ. Unidades: IFSC, ICB
Subjects: MALÁRIA, PLASMODIUM FALCIPARUM, PLANEJAMENTO DE FÁRMACOS
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ABNT
OLIVEIRA, Douglas Davison da Silva et al. Hit-to-Lead optimization of pyridylpiperazine derivatives: promising antimalarial candidates with notable ADME profiles and metabolic stability. 2025, Anais.. São Paulo: Sociedade Brasileira de Química - SBQ, 2025. Disponível em: https://repositorio.usp.br/directbitstream/f179559b-b0ab-49da-8d2d-69b170cab755/3259728.pdf. Acesso em: 08 out. 2025.
APA
Oliveira, D. D. da S., Krüger, A., Chelucci, R. C., Ferreira, L. L. G., Andricopulo, A. D., Wunderlich, G., et al. (2025). Hit-to-Lead optimization of pyridylpiperazine derivatives: promising antimalarial candidates with notable ADME profiles and metabolic stability. In Anais. São Paulo: Sociedade Brasileira de Química - SBQ. Recuperado de https://repositorio.usp.br/directbitstream/f179559b-b0ab-49da-8d2d-69b170cab755/3259728.pdf
NLM
Oliveira DD da S, Krüger A, Chelucci RC, Ferreira LLG, Andricopulo AD, Wunderlich G, Silva NM da, Rezende Junior C de O. Hit-to-Lead optimization of pyridylpiperazine derivatives: promising antimalarial candidates with notable ADME profiles and metabolic stability [Internet]. Anais. 2025 ;[citado 2025 out. 08 ] Available from: https://repositorio.usp.br/directbitstream/f179559b-b0ab-49da-8d2d-69b170cab755/3259728.pdf
Vancouver
Oliveira DD da S, Krüger A, Chelucci RC, Ferreira LLG, Andricopulo AD, Wunderlich G, Silva NM da, Rezende Junior C de O. Hit-to-Lead optimization of pyridylpiperazine derivatives: promising antimalarial candidates with notable ADME profiles and metabolic stability [Internet]. Anais. 2025 ;[citado 2025 out. 08 ] Available from: https://repositorio.usp.br/directbitstream/f179559b-b0ab-49da-8d2d-69b170cab755/3259728.pdf
Artigo de periodico
Hit-to-lead studies of pyrazinylpiperazines against visceral Leishmaniasis: pharmacokinetic profile and in vivo efficacy of potent compounds against Leishmania infantum (2025)
Lapierre, Thibault Joseph William Jacques Dit ; Cruz, Mariza Gabriela Faleiro de Moura Lodi; Barbosa, Gisele; Costa, Analu Rocha ; Chávez-Fumagalli, Miguel Angel ; Froes, Thamires Quadros ; Ramos, Priscila Zonzini; Macruz, Paula Derksen; Trindade, Thalita Carolyne Souza; Pilau, Eduardo Jorge ; Veras, Patricia Sampaio Tavares; Nonato, Maria Cristina ; Massirer, Katlin Brauer ; Ferreira, Leonardo Luiz Gomes ; Andricopulo, Adriano Defini ; Lima, Lídia Moreira ; Murta, Silvane Maria Fonseca ; Rezende Junior, Celso de Oliveira
Source: ACS Pharmacology and Translational Science. Unidades: FCFRP, IFSC
Subjects: LEISHMANIA, CRISTALOGRAFIA, FÁRMACOS
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ABNT
LAPIERRE, Thibault Joseph William Jacques Dit et al. Hit-to-lead studies of pyrazinylpiperazines against visceral Leishmaniasis: pharmacokinetic profile and in vivo efficacy of potent compounds against Leishmania infantum. ACS Pharmacology and Translational Science, v. 8, n. 8, p. 2736–2755 + supporting information, 2025Tradução . . Disponível em: https://doi.org/10.1021/acsptsci.5c00318. Acesso em: 08 out. 2025.
APA
Lapierre, T. J. W. J. D., Cruz, M. G. F. de M. L., Barbosa, G., Costa, A. R., Chávez-Fumagalli, M. A., Froes, T. Q., et al. (2025). Hit-to-lead studies of pyrazinylpiperazines against visceral Leishmaniasis: pharmacokinetic profile and in vivo efficacy of potent compounds against Leishmania infantum. ACS Pharmacology and Translational Science, 8( 8), 2736–2755 + supporting information. doi:10.1021/acsptsci.5c00318
NLM
Lapierre TJWJD, Cruz MGF de ML, Barbosa G, Costa AR, Chávez-Fumagalli MA, Froes TQ, Ramos PZ, Macruz PD, Trindade TCS, Pilau EJ, Veras PST, Nonato MC, Massirer KB, Ferreira LLG, Andricopulo AD, Lima LM, Murta SMF, Rezende Junior C de O. Hit-to-lead studies of pyrazinylpiperazines against visceral Leishmaniasis: pharmacokinetic profile and in vivo efficacy of potent compounds against Leishmania infantum [Internet]. ACS Pharmacology and Translational Science. 2025 ; 8( 8): 2736–2755 + supporting information.[citado 2025 out. 08 ] Available from: https://doi.org/10.1021/acsptsci.5c00318
Vancouver
Lapierre TJWJD, Cruz MGF de ML, Barbosa G, Costa AR, Chávez-Fumagalli MA, Froes TQ, Ramos PZ, Macruz PD, Trindade TCS, Pilau EJ, Veras PST, Nonato MC, Massirer KB, Ferreira LLG, Andricopulo AD, Lima LM, Murta SMF, Rezende Junior C de O. Hit-to-lead studies of pyrazinylpiperazines against visceral Leishmaniasis: pharmacokinetic profile and in vivo efficacy of potent compounds against Leishmania infantum [Internet]. ACS Pharmacology and Translational Science. 2025 ; 8( 8): 2736–2755 + supporting information.[citado 2025 out. 08 ] Available from: https://doi.org/10.1021/acsptsci.5c00318
Artigo de periodico
Discovery of arylpiperazines with broad-spectrum antimicrobial activity and favorable pharmacokinetic profiles (2025)
Oliveira, Douglas Davison da Silva ; Silva, Nagela Bernadelli Sousa; Lapierre, Thibault Joseph William Jacques Dit ; Souza, Sara Lemes de; Brito, Nícolas Peterson Ferreira ; Martinho, Ana Clara Cassiano ; Dias, Renieidy Flávia Clemente; Farago, Danilo Nascimento; Duarte, Simone Michelan ; Chelucci, Rafael Consolin; Cruz, Mariza Gabriela Faleiro de Moura Lodi; Resende, Daniela de Melo ; Andricopulo, Adriano Defini ; Murta, Silvane Maria Fonseca ; Ferreira, Leonardo Luiz Gomes ; Martins, Carlos Henrique Gomes ; Rezende Junior, Celso de Oliveira
Source: Chemistry and Biodiversity. Unidade: IFSC
Subjects: PLANEJAMENTO DE FÁRMACOS, RESISTÊNCIA MICROBIANA ÀS DROGAS, CITOTOXINAS
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ABNT
OLIVEIRA, Douglas Davison da Silva et al. Discovery of arylpiperazines with broad-spectrum antimicrobial activity and favorable pharmacokinetic profiles. Chemistry and Biodiversity, v. 22, n. 2, p. e202402100-1-e202402100-14, 2025Tradução . . Disponível em: https://doi.org/10.1002/cbdv.202402100. Acesso em: 08 out. 2025.
APA
Oliveira, D. D. da S., Silva, N. B. S., Lapierre, T. J. W. J. D., Souza, S. L. de, Brito, N. P. F., Martinho, A. C. C., et al. (2025). Discovery of arylpiperazines with broad-spectrum antimicrobial activity and favorable pharmacokinetic profiles. Chemistry and Biodiversity, 22( 2), e202402100-1-e202402100-14. doi:10.1002/cbdv.202402100
NLM
Oliveira DD da S, Silva NBS, Lapierre TJWJD, Souza SL de, Brito NPF, Martinho ACC, Dias RFC, Farago DN, Duarte SM, Chelucci RC, Cruz MGF de ML, Resende D de M, Andricopulo AD, Murta SMF, Ferreira LLG, Martins CHG, Rezende Junior C de O. Discovery of arylpiperazines with broad-spectrum antimicrobial activity and favorable pharmacokinetic profiles [Internet]. Chemistry and Biodiversity. 2025 ; 22( 2): e202402100-1-e202402100-14.[citado 2025 out. 08 ] Available from: https://doi.org/10.1002/cbdv.202402100
Vancouver
Oliveira DD da S, Silva NBS, Lapierre TJWJD, Souza SL de, Brito NPF, Martinho ACC, Dias RFC, Farago DN, Duarte SM, Chelucci RC, Cruz MGF de ML, Resende D de M, Andricopulo AD, Murta SMF, Ferreira LLG, Martins CHG, Rezende Junior C de O. Discovery of arylpiperazines with broad-spectrum antimicrobial activity and favorable pharmacokinetic profiles [Internet]. Chemistry and Biodiversity. 2025 ; 22( 2): e202402100-1-e202402100-14.[citado 2025 out. 08 ] Available from: https://doi.org/10.1002/cbdv.202402100
Artigo de periodico
Machine learning-based virtual screening of antibacterial agents against methicillin-susceptible and resistant staphylococcus aureus (2024)
Fernandes, Philipe Oliveira ; Dias, Anna Letícia Teotonio; Santos Júnior, Valtair Severino dos ; Serafim, Mateus Sá Magalhães ; Sousa, Yamara Viana; Monteiro, Gustavo Claro ; Coutinho, Isabel Duarte ; Valli, Marilia ; Verzola, Marina Mol Sena Andrade; Ottoni, Flaviano Melo; Pádua, Rodrigo Maia de; Oda, Fernando Bombarda ; Santos, André Gonzaga dos ; Andricopulo, Adriano Defini ; Bolzani, Vanderlan da Silva ; Mota, Bruno Eduardo Fernandes; Alves, Ricardo José; Oliveira, Renata Barbosa de ; Kronenberger, Thales ; Maltarollo, Vinícius Gonçalves
Source: Journal of Chemical Information and Modeling. Unidade: IFSC
Subjects: BACTÉRIAS, AGENTES ANTIMICROBIANOS, CRISTALOGRAFIA
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ABNT
FERNANDES, Philipe Oliveira et al. Machine learning-based virtual screening of antibacterial agents against methicillin-susceptible and resistant staphylococcus aureus. Journal of Chemical Information and Modeling, v. 64, n. 6, p. 1932-1944 + supporting information, 2024Tradução . . Disponível em: https://doi.org/10.1021/acs.jcim.4c00087. Acesso em: 08 out. 2025.
APA
Fernandes, P. O., Dias, A. L. T., Santos Júnior, V. S. dos, Serafim, M. S. M., Sousa, Y. V., Monteiro, G. C., et al. (2024). Machine learning-based virtual screening of antibacterial agents against methicillin-susceptible and resistant staphylococcus aureus. Journal of Chemical Information and Modeling, 64( 6), 1932-1944 + supporting information. doi:10.1021/acs.jcim.4c00087
NLM
Fernandes PO, Dias ALT, Santos Júnior VS dos, Serafim MSM, Sousa YV, Monteiro GC, Coutinho ID, Valli M, Verzola MMSA, Ottoni FM, Pádua RM de, Oda FB, Santos AG dos, Andricopulo AD, Bolzani V da S, Mota BEF, Alves RJ, Oliveira RB de, Kronenberger T, Maltarollo VG. Machine learning-based virtual screening of antibacterial agents against methicillin-susceptible and resistant staphylococcus aureus [Internet]. Journal of Chemical Information and Modeling. 2024 ; 64( 6): 1932-1944 + supporting information.[citado 2025 out. 08 ] Available from: https://doi.org/10.1021/acs.jcim.4c00087
Vancouver
Fernandes PO, Dias ALT, Santos Júnior VS dos, Serafim MSM, Sousa YV, Monteiro GC, Coutinho ID, Valli M, Verzola MMSA, Ottoni FM, Pádua RM de, Oda FB, Santos AG dos, Andricopulo AD, Bolzani V da S, Mota BEF, Alves RJ, Oliveira RB de, Kronenberger T, Maltarollo VG. Machine learning-based virtual screening of antibacterial agents against methicillin-susceptible and resistant staphylococcus aureus [Internet]. Journal of Chemical Information and Modeling. 2024 ; 64( 6): 1932-1944 + supporting information.[citado 2025 out. 08 ] Available from: https://doi.org/10.1021/acs.jcim.4c00087
Artigo de periodico
Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum (2024)
Lapierre, Thibault Joseph William Jacques Dit ; Farago, Danilo Nascimento; Cruz, Mariza Gabriela Faleiro de Moura Lodi; Resende, Daniela de Melo ; Oliveira, Adriane Cristina Rosa de; Santos, Brenda Rosa Macedo dos; Souza, Felipe de Oliveira; Duarte, Simone Michelan ; Chelucci, Rafael Consolin; Andricopulo, Adriano Defini ; Ferreira, Leonardo Luiz Gomes ; Pilau, Eduardo Jorge ; Murta, Silvane Maria Fonseca ; Rezende Junior, Celso de Oliveira
Source: Chemical Biology and Drug Design. Unidade: IFSC
Subjects: LEISHMANIA, MECANISMOS DE DEFESA, TRYPANOSOMA CRUZI
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ABNT
LAPIERRE, Thibault Joseph William Jacques Dit et al. Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum. Chemical Biology and Drug Design, v. 103, p. e14525-1-e14525-14 + supporting information, 2024Tradução . . Disponível em: https://doi.org/10.1111/cbdd.14525. Acesso em: 08 out. 2025.
APA
Lapierre, T. J. W. J. D., Farago, D. N., Cruz, M. G. F. de M. L., Resende, D. de M., Oliveira, A. C. R. de, Santos, B. R. M. dos, et al. (2024). Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum. Chemical Biology and Drug Design, 103, e14525-1-e14525-14 + supporting information. doi:10.1111/cbdd.14525
NLM
Lapierre TJWJD, Farago DN, Cruz MGF de ML, Resende D de M, Oliveira ACR de, Santos BRM dos, Souza F de O, Duarte SM, Chelucci RC, Andricopulo AD, Ferreira LLG, Pilau EJ, Murta SMF, Rezende Junior C de O. Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum [Internet]. Chemical Biology and Drug Design. 2024 ; 103 e14525-1-e14525-14 + supporting information.[citado 2025 out. 08 ] Available from: https://doi.org/10.1111/cbdd.14525
Vancouver
Lapierre TJWJD, Farago DN, Cruz MGF de ML, Resende D de M, Oliveira ACR de, Santos BRM dos, Souza F de O, Duarte SM, Chelucci RC, Andricopulo AD, Ferreira LLG, Pilau EJ, Murta SMF, Rezende Junior C de O. Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum [Internet]. Chemical Biology and Drug Design. 2024 ; 103 e14525-1-e14525-14 + supporting information.[citado 2025 out. 08 ] Available from: https://doi.org/10.1111/cbdd.14525

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