Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor (2020)
- Authors:
- USP affiliated authors: LEITÃO, ANDREI - IQSC ; MONTANARI, CARLOS ALBERTO - IQSC ; ROSINI, FABIANA - IQSC ; RIBEIRO, JEAN FRANCISCO ROSA - IQSC ; CIANNI, LORENZO - IQSC ; VITA, DANIELA DE - IQSC ; ROCHO, FERNANDA DOS REIS - IQSC ; MARTINS, FELIPE CARDOSO PRADO - IQSC
- Unidade: IQSC
- DOI: 10.1016/j.bmc.2020.115743
- Subjects: LEISHMANIA MEXICANA; MEDICAMENTO
- Keywords: Crystal structure; Leishmania mexicana cysteine protease B; Azadipeptide nitrile inhibitor; Structure activity relationships (SARs); Covalent inhibitor
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Source:
- Título: Bioorganic and Medicinal Chemistry
- ISSN: 0968-0896
- Volume/Número/Paginação/Ano: v. 22, n. 22, p. 115743, November 2020
- Este periódico é de assinatura
- Este artigo NÃO é de acesso aberto
- Cor do Acesso Aberto: closed
-
ABNT
RIBEIRO, Jean Francisco Rosa et al. Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor. Bioorganic and Medicinal Chemistry, v. 22, n. 22, p. 115743, 2020Tradução . . Disponível em: https://doi.org/10.1016/j.bmc.2020.115743. Acesso em: 27 dez. 2025. -
APA
Ribeiro, J. F. R., Cianni, L., Li, C., Warwick, T. G., Vita, D. de, Rosini, F., et al. (2020). Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor. Bioorganic and Medicinal Chemistry, 22( 22), 115743. doi:10.1016/j.bmc.2020.115743 -
NLM
Ribeiro JFR, Cianni L, Li C, Warwick TG, Vita D de, Rosini F, Rocho F dos R, Martins FCP, Kenny PW, Lameira J, Leitão A, Emsley J, Montanari CA. Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor [Internet]. Bioorganic and Medicinal Chemistry. 2020 ; 22( 22): 115743.[citado 2025 dez. 27 ] Available from: https://doi.org/10.1016/j.bmc.2020.115743 -
Vancouver
Ribeiro JFR, Cianni L, Li C, Warwick TG, Vita D de, Rosini F, Rocho F dos R, Martins FCP, Kenny PW, Lameira J, Leitão A, Emsley J, Montanari CA. Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor [Internet]. Bioorganic and Medicinal Chemistry. 2020 ; 22( 22): 115743.[citado 2025 dez. 27 ] Available from: https://doi.org/10.1016/j.bmc.2020.115743 - N-Sulfonyl dipeptide nitriles as inhibitors of human cathepsin S: In silico design, synthesis and biochemical characterization
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Informações sobre o DOI: 10.1016/j.bmc.2020.115743 (Fonte: oaDOI API)
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