Synthesis and optimization of indole-2-carboxamides for enhanced anti-plasmodial activity (2025)
- Authors:
- USP affiliated authors: GUIDO, RAFAEL VICTÓRIO CARVALHO - IFSC ; AGUIAR, ANNA CAROLINE CAMPOS - IFSC ; MALUF, SARAH EL CHAMY - IFSC
- Unidade: IFSC
- Subjects: PROTEÍNAS; MALÁRIA; ANTIMALÁRICOS; CRISTALOGRAFIA; PLANEJAMENTO DE FÁRMACOS
- Keywords: Malaria; Indoles; Carboxamides; Chloroquine; SAR studies; Cross-resistance
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Publisher: Universidade Federal do Rio de Janeiro - UFRJ
- Publisher place: Rio de Janeiro
- Date published: 2025
- Source:
- Título: Annals
- Conference titles: Brazilian Symposium on Medicinal Chemistry - BrazMedChem
-
ABNT
CARMELLO, Stephany Vieira et al. Synthesis and optimization of indole-2-carboxamides for enhanced anti-plasmodial activity. 2025, Anais.. Rio de Janeiro: Universidade Federal do Rio de Janeiro - UFRJ, 2025. Disponível em: https://repositorio.usp.br/directbitstream/4b7b3a18-2460-46b4-a90d-7ea3f8deae16/PROD038180_3290864.pdf. Acesso em: 30 mar. 2026. -
APA
Carmello, S. V., Sacchelli, B. A. L., Ahmad, A., Kumar , M., Aguiar, A. C. C., Maluf, S. E. C., et al. (2025). Synthesis and optimization of indole-2-carboxamides for enhanced anti-plasmodial activity. In Annals. Rio de Janeiro: Universidade Federal do Rio de Janeiro - UFRJ. Recuperado de https://repositorio.usp.br/directbitstream/4b7b3a18-2460-46b4-a90d-7ea3f8deae16/PROD038180_3290864.pdf -
NLM
Carmello SV, Sacchelli BAL, Ahmad A, Kumar M, Aguiar ACC, Maluf SEC, Shamim A, Ferrer MC, Geldern TW von, Baud D, Jones B, Willis PA, Duffy J, Guido RVC, Dias LC. Synthesis and optimization of indole-2-carboxamides for enhanced anti-plasmodial activity [Internet]. Annals. 2025 ;[citado 2026 mar. 30 ] Available from: https://repositorio.usp.br/directbitstream/4b7b3a18-2460-46b4-a90d-7ea3f8deae16/PROD038180_3290864.pdf -
Vancouver
Carmello SV, Sacchelli BAL, Ahmad A, Kumar M, Aguiar ACC, Maluf SEC, Shamim A, Ferrer MC, Geldern TW von, Baud D, Jones B, Willis PA, Duffy J, Guido RVC, Dias LC. Synthesis and optimization of indole-2-carboxamides for enhanced anti-plasmodial activity [Internet]. Annals. 2025 ;[citado 2026 mar. 30 ] Available from: https://repositorio.usp.br/directbitstream/4b7b3a18-2460-46b4-a90d-7ea3f8deae16/PROD038180_3290864.pdf - Multiparametric optimization of pyrazole compounds with antimalarial activity
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