Optimization of compounds from the pyrazole series for malaria treatment (2025)
- Authors:
- USP affiliated authors: GUIDO, RAFAEL VICTÓRIO CARVALHO - IFSC ; MALUF, SARAH EL CHAMY - IFSC ; SOUZA, GUILHERME EDUARDO DE - IFSC ; AGUIAR, ANNA CAROLINE CAMPOS - IFSC
- Unidade: IFSC
- Subjects: PLANEJAMENTO DE FÁRMACOS; MALÁRIA; CRISTALOGRAFIA
- Keywords: Drug discovery; Malaria; Organic chemistry; Synthesis; SAR; Pyrazole
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Publisher: Sociedade Brasileira de Química - SBQ
- Publisher place: São Paulo
- Date published: 2025
- Source:
- Título: Anais
- Conference titles: Reunião Anual da Sociedade Brasileira de Química - RASBQ
-
ABNT
CARMELLO, Stephany Vieira et al. Optimization of compounds from the pyrazole series for malaria treatment. 2025, Anais.. São Paulo: Sociedade Brasileira de Química - SBQ, 2025. Disponível em: https://repositorio.usp.br/directbitstream/4b1e5496-7e47-42b0-a138-0fe2b38dc9f6/3259925.pdf. Acesso em: 30 mar. 2026. -
APA
Carmello, S. V., Okada Júnior, C. Y., Kumar, M., Casal, M. F., Ahmad, A., Shamim, A., et al. (2025). Optimization of compounds from the pyrazole series for malaria treatment. In Anais. São Paulo: Sociedade Brasileira de Química - SBQ. Recuperado de https://repositorio.usp.br/directbitstream/4b1e5496-7e47-42b0-a138-0fe2b38dc9f6/3259925.pdf -
NLM
Carmello SV, Okada Júnior CY, Kumar M, Casal MF, Ahmad A, Shamim A, Maluf SEC, Souza GE de, Aguiar ACC, Guido RVC, Geldern T von, Baud D, Willis P, Jones B, Dias LC. Optimization of compounds from the pyrazole series for malaria treatment [Internet]. Anais. 2025 ;[citado 2026 mar. 30 ] Available from: https://repositorio.usp.br/directbitstream/4b1e5496-7e47-42b0-a138-0fe2b38dc9f6/3259925.pdf -
Vancouver
Carmello SV, Okada Júnior CY, Kumar M, Casal MF, Ahmad A, Shamim A, Maluf SEC, Souza GE de, Aguiar ACC, Guido RVC, Geldern T von, Baud D, Willis P, Jones B, Dias LC. Optimization of compounds from the pyrazole series for malaria treatment [Internet]. Anais. 2025 ;[citado 2026 mar. 30 ] Available from: https://repositorio.usp.br/directbitstream/4b1e5496-7e47-42b0-a138-0fe2b38dc9f6/3259925.pdf - Indole-2-carboxamides optimization for antiplasmodial activity
- MMV's drug discovery project: test cascade towards the development of new antimalarials
- Synthesis and optimization of indole-2-carboxamides for enhanced anti-plasmodial activity
- Multiparametric optimization of pyrazole compounds with antimalarial activity
- Development of a structure-activity relationship study for the Thiadiazole series
- Thiadiazole derived compounds as new Plasmodium falciparum inhibitors: synthesis and structure-activity relationships
- Descoberta de derivados de marinoquinolina como inibidores de Plasmodium falciparum
- Marinoquinolines as highly active and selective antimalarial compounds
- Estudo do efeito de um grupo espaçador metilênico em marinoquinolinas: síntese e avaliação biológica
- Descoberta de derivados de marinoquinolina como inibidores de Plasmodium falciparum
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