Pyrimidine azepine targets the plasmodium bc1 complex and displays multistage antimalarial activit (2024)
- Authors:
- Calit, Juliana

- Prajapati , Surendra K.
- Benavente, Ernest Diez

- Araújo, Jéssica Evangelista
- Deng, Bingbing

- Miura, Kazutoyo

- Annunciato, Yasmin

- Moura, Igor Mota Rodrigues de

- Usui, Miho
- Medeiros, Jansen Fernandes de

- Andrade, Carolina Horta

- Mendonça, Sabrina Silva
- Simeonov, Anton
- Eastman, Richard T.

- Long, Carole A.

- Araújo, Maisa da Silva

- Williamson, Kim C.

- Aguiar, Anna Caroline Campos

- Bargieri, Daniel Youssef

- Calit, Juliana
- USP affiliated authors: BARGIERI, DANIEL YOUSSEF - ICB ; PAIM, JULIANA CALIT - ICB ; MOURA, IGOR MOTA RODRIGUES DE - IFSC
- Unidades: ICB; IFSC
- DOI: 10.1021/jacsau.4c00674
- Subjects: MALÁRIA; PLANEJAMENTO DE FÁRMACOS; PLASMODIUM FALCIPARUM; ANTIMALÁRICOS
- Keywords: Malaria; Resistance; Pyrimidine azepine; Bc1 complex; Plasmodium
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Publisher place: Washington, DC
- Date published: 2024
- Source:
- Status:
- Artigo publicado em periódico de acesso aberto (Gold Open Access)
- Versão do Documento:
- Versão publicada (Published version)
- Acessar versão aberta:
-
ABNT
CALIT, Juliana et al. Pyrimidine azepine targets the plasmodium bc1 complex and displays multistage antimalarial activit. JACS Au, v. 4, n. 10, p. 3942-3952 + supporting information, 2024Tradução . . Disponível em: https://doi.org/10.1021/jacsau.4c00674. Acesso em: 31 mar. 2026. -
APA
Calit, J., Prajapati , S. K., Benavente, E. D., Araújo, J. E., Deng, B., Miura, K., et al. (2024). Pyrimidine azepine targets the plasmodium bc1 complex and displays multistage antimalarial activit. JACS Au, 4( 10), 3942-3952 + supporting information. doi:10.1021/jacsau.4c00674 -
NLM
Calit J, Prajapati SK, Benavente ED, Araújo JE, Deng B, Miura K, Annunciato Y, Moura IMR de, Usui M, Medeiros JF de, Andrade CH, Mendonça SS, Simeonov A, Eastman RT, Long CA, Araújo M da S, Williamson KC, Aguiar ACC, Bargieri DY. Pyrimidine azepine targets the plasmodium bc1 complex and displays multistage antimalarial activit [Internet]. JACS Au. 2024 ; 4( 10): 3942-3952 + supporting information.[citado 2026 mar. 31 ] Available from: https://doi.org/10.1021/jacsau.4c00674 -
Vancouver
Calit J, Prajapati SK, Benavente ED, Araújo JE, Deng B, Miura K, Annunciato Y, Moura IMR de, Usui M, Medeiros JF de, Andrade CH, Mendonça SS, Simeonov A, Eastman RT, Long CA, Araújo M da S, Williamson KC, Aguiar ACC, Bargieri DY. Pyrimidine azepine targets the plasmodium bc1 complex and displays multistage antimalarial activit [Internet]. JACS Au. 2024 ; 4( 10): 3942-3952 + supporting information.[citado 2026 mar. 31 ] Available from: https://doi.org/10.1021/jacsau.4c00674 - Computational chemogenomics drug repositioning strategy enables the discovery of epirubicin as a new repurposed hit for Plasmodium Falciparum and P. vivax
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