Novel selective proline-based peptidomimetics for human cathepsin K inhibition (2024)
- Authors:
- USP affiliated authors: LEITÃO, ANDREI - IQSC ; MONTANARI, CARLOS ALBERTO - IQSC ; MARTINS, FELIPE CARDOSO PRADO - IQSC ; ROCHO, FERNANDA DOS REIS - IQSC ; BONATTO, VINÍCIUS - IQSC ; BATISTA, PEDRO HENRIQUE JATAI - IQSC
- Unidade: IQSC
- DOI: 10.1016/j.bmcl.2024.129887
- Subjects: INIBIDORES QUÍMICOS; OSTEOPOROSE
- Keywords: Cysteine protease; Human cathepsin K; Nitrile inhibitors; Rigid analog
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Source:
- Título: Bioorganic & Medicinal Chemistry Letters
- ISSN: 1464-3405
- Volume/Número/Paginação/Ano: v.110, p.129887, 2024
- Este periódico é de assinatura
- Este artigo NÃO é de acesso aberto
- Cor do Acesso Aberto: closed
-
ABNT
MARTINS, Felipe Cardoso Prado et al. Novel selective proline-based peptidomimetics for human cathepsin K inhibition. Bioorganic & Medicinal Chemistry Letters, v. 110, p. 129887, 2024Tradução . . Disponível em: https://doi.org/10.1016/j.bmcl.2024.129887. Acesso em: 27 dez. 2025. -
APA
Martins, F. C. P., Rocho, F. dos R., Bonatto, V., Batista, P. H. J., Lameira, J., Leitão, A., & Montanari, C. A. (2024). Novel selective proline-based peptidomimetics for human cathepsin K inhibition. Bioorganic & Medicinal Chemistry Letters, 110, 129887. doi:10.1016/j.bmcl.2024.129887 -
NLM
Martins FCP, Rocho F dos R, Bonatto V, Batista PHJ, Lameira J, Leitão A, Montanari CA. Novel selective proline-based peptidomimetics for human cathepsin K inhibition [Internet]. Bioorganic & Medicinal Chemistry Letters. 2024 ;110 129887.[citado 2025 dez. 27 ] Available from: https://doi.org/10.1016/j.bmcl.2024.129887 -
Vancouver
Martins FCP, Rocho F dos R, Bonatto V, Batista PHJ, Lameira J, Leitão A, Montanari CA. Novel selective proline-based peptidomimetics for human cathepsin K inhibition [Internet]. Bioorganic & Medicinal Chemistry Letters. 2024 ;110 129887.[citado 2025 dez. 27 ] Available from: https://doi.org/10.1016/j.bmcl.2024.129887 - Exploring Nirmatrelvir derivatives through P2 substituent modifications and warhead innovations targeting the main protease of SARS-CoV-2
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Informações sobre o DOI: 10.1016/j.bmcl.2024.129887 (Fonte: oaDOI API)
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