Using a fragment-based approach to identify alternative chemical scaffolds targeting dihydrofolate reductase from Mycobacterium tuberculosis (2020)
- Authors:
- Ribeiro, João A.
- Hammer, Alexander
- Zuniga, Gerardo A. Libreros
- Pacheco, Sair Maximo Chavez
- Tyrakis, Petros
- Oliveira, Gabriel S. de
- Kirkman, Timothy
- Bakali, Jamal El
- Rocco, Silvana A.
- Sforça, Mauricio L.
- Parise Filho, Roberto
- Coyne, Anthony G.
- Blundell, Tom L.
- Abell, Chris
- Dias, Marcio Vinicius Bertacine
- USP affiliated authors: PARISE FILHO, ROBERTO - FCF ; DIAS, MARCIO VINÍCIUS BERTACINE - ICB
- Unidades: FCF; ICB
- DOI: 10.1021/acsinfecdis.0c00263
- Subjects: MYCOBACTERIUM TUBERCULOSIS; ÁCIDO FÓLICO; MICROBIOLOGIA; INIBIDORES DE ENZIMAS; ATIVAÇÃO ENZIMÁTICA
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Publisher place: Washington
- Date published: 2020
- Source:
- Título: ACS Infectious Diseases
- ISSN: 2373-8227
- Volume/Número/Paginação/Ano: v. 6, p. 2192−2201 : + Supplementary materials (p. S1-S16), 2020
- Este periódico é de acesso aberto
- Este artigo NÃO é de acesso aberto
-
ABNT
RIBEIRO, João A. et al. Using a fragment-based approach to identify alternative chemical scaffolds targeting dihydrofolate reductase from Mycobacterium tuberculosis. ACS Infectious Diseases, v. 6, p. 2192−2201 : + Supplementary materials ( S1-S16), 2020Tradução . . Disponível em: https://doi.org/10.1021/acsinfecdis.0c00263. Acesso em: 10 fev. 2026. -
APA
Ribeiro, J. A., Hammer, A., Zuniga, G. A. L., Pacheco, S. M. C., Tyrakis, P., Oliveira, G. S. de, et al. (2020). Using a fragment-based approach to identify alternative chemical scaffolds targeting dihydrofolate reductase from Mycobacterium tuberculosis. ACS Infectious Diseases, 6, 2192−2201 : + Supplementary materials ( S1-S16). doi:10.1021/acsinfecdis.0c00263 -
NLM
Ribeiro JA, Hammer A, Zuniga GAL, Pacheco SMC, Tyrakis P, Oliveira GS de, Kirkman T, Bakali JE, Rocco SA, Sforça ML, Parise Filho R, Coyne AG, Blundell TL, Abell C, Dias MVB. Using a fragment-based approach to identify alternative chemical scaffolds targeting dihydrofolate reductase from Mycobacterium tuberculosis [Internet]. ACS Infectious Diseases. 2020 ; 6 2192−2201 : + Supplementary materials ( S1-S16).[citado 2026 fev. 10 ] Available from: https://doi.org/10.1021/acsinfecdis.0c00263 -
Vancouver
Ribeiro JA, Hammer A, Zuniga GAL, Pacheco SMC, Tyrakis P, Oliveira GS de, Kirkman T, Bakali JE, Rocco SA, Sforça ML, Parise Filho R, Coyne AG, Blundell TL, Abell C, Dias MVB. Using a fragment-based approach to identify alternative chemical scaffolds targeting dihydrofolate reductase from Mycobacterium tuberculosis [Internet]. ACS Infectious Diseases. 2020 ; 6 2192−2201 : + Supplementary materials ( S1-S16).[citado 2026 fev. 10 ] Available from: https://doi.org/10.1021/acsinfecdis.0c00263 - Optimization of new dihydrofolate reductase inhibitors of mycobacterium tuberculosis (mtDHFR): molecular docking, synthesis, evaluation of enzyme inhibition and antimycobacterial activity
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Informações sobre o DOI: 10.1021/acsinfecdis.0c00263 (Fonte: oaDOI API)
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