Artigo de periodico

Structure-based and molecular modeling studies for the discovery of cyclic imides as reversible cruzain inhibitors with potent anti-Trypanosoma cruzi activity (2019)

• Authors:
  • Ferreira, Rafael A. A.
  • Pauli, Ivani
  • Sampaio, Thiago S.
  • Souza, Mariana Laureano de
  • Ferreira, Leonardo Luiz Gomes
  • Magalhães, Luma Godoy
  • Rezende Junior, Celso O.
  • Ferreira, Rafaela S.
  • Krogh, Renata
  • Dias, Luiz C.
  • Andricopulo, Adriano Defini
• USP affiliated authors: ANDRICOPULO, RENATA KROGH - IFSC ; ANDRICOPULO, ADRIANO DEFINI - IFSC ; PAULI, IVANÍ - IFSC ; SOUZA, MARIANA LAUREANO DE - IFSC ; FERREIRA, LEONARDO LUIZ GOMES - IFSC ; MAGALHÃES, LUMA GODOY - IFSC
• Unidade: IFSC
• DOI: 10.3389/fchem.2019.00798
• Subjects: DOENÇA DE CHAGAS; TRYPANOSOMA CRUZI; PLANEJAMENTO DE FÁRMACOS
• Keywords: Chagas disease; Trypanosoma cruzi; Cruzain; SAR; Medicinal chemistry; Synthesis; Inhibitors; Molecular docking
• Agências de fomento:
  • Financiado pelo CNPq
  • Financiado pela CAPES
  • Financiado pela FAPESP
• Language: Inglês
• Imprenta:
  • Publisher place: Lausanne
  • Date published: 2019
• Source:
  • Título: Frontiers in Chemistry
  • ISSN: 2296-2646
  • Volume/Número/Paginação/Ano: v. 7, p. 798-1-798-21, Nov. 2019


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• ABNT

  FERREIRA, Rafael A. A. et al. Structure-based and molecular modeling studies for the discovery of cyclic imides as reversible cruzain inhibitors with potent anti-Trypanosoma cruzi activity. Frontiers in Chemistry, v. No 2019, p. 798-1-798-21, 2019Tradução . . Disponível em: https://doi.org/10.3389/fchem.2019.00798. Acesso em: 01 abr. 2026.

• APA

  Ferreira, R. A. A., Pauli, I., Sampaio, T. S., Souza, M. L. de, Ferreira, L. L. G., Magalhães, L. G., et al. (2019). Structure-based and molecular modeling studies for the discovery of cyclic imides as reversible cruzain inhibitors with potent anti-Trypanosoma cruzi activity. Frontiers in Chemistry, No 2019, 798-1-798-21. doi:10.3389/fchem.2019.00798

• NLM

  Ferreira RAA, Pauli I, Sampaio TS, Souza ML de, Ferreira LLG, Magalhães LG, Rezende Junior CO, Ferreira RS, Krogh R, Dias LC, Andricopulo AD. Structure-based and molecular modeling studies for the discovery of cyclic imides as reversible cruzain inhibitors with potent anti-Trypanosoma cruzi activity [Internet]. Frontiers in Chemistry. 2019 ; No 2019 798-1-798-21.[citado 2026 abr. 01 ] Available from: https://doi.org/10.3389/fchem.2019.00798

• Vancouver

  Ferreira RAA, Pauli I, Sampaio TS, Souza ML de, Ferreira LLG, Magalhães LG, Rezende Junior CO, Ferreira RS, Krogh R, Dias LC, Andricopulo AD. Structure-based and molecular modeling studies for the discovery of cyclic imides as reversible cruzain inhibitors with potent anti-Trypanosoma cruzi activity [Internet]. Frontiers in Chemistry. 2019 ; No 2019 798-1-798-21.[citado 2026 abr. 01 ] Available from: https://doi.org/10.3389/fchem.2019.00798

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