Brazilian Symposium on Medicinal Chemistry - BrazMedChem, 11 (2023)
- Autores:
- Autores USP: ANDRICOPULO, ADRIANO DEFINI - IFSC ; TROSSINI, GUSTAVO HENRIQUE GOULART - FCF ; NONATO, MARIA CRISTINA - FCFRP ; NASCIMENTO, ALESSANDRO SILVA - IFSC ; EMERY, FLAVIO DA SILVA - FCFRP ; DIAS, MARCIO VINÍCIUS BERTACINE - ICB ; PARISE FILHO, ROBERTO - FCF
- Unidades: IFSC; FCF; FCFRP; ICB
- Assuntos: CRISTALOGRAFIA; QUÍMICA MÉDICA; PESQUISA CIENTÍFICA
- Idioma: Inglês
- Imprenta:
- Editora: Universidade Federal da Bahia - UFBA
- Local: Salvador
- Data de publicação: 2023
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ABNT
Brazilian Symposium on Medicinal Chemistry - BrazMedChem, 11. . Salvador: Universidade Federal da Bahia - UFBA. . Acesso em: 02 out. 2024. , 2023 -
APA
Brazilian Symposium on Medicinal Chemistry - BrazMedChem, 11. (2023). Brazilian Symposium on Medicinal Chemistry - BrazMedChem, 11. Salvador: Universidade Federal da Bahia - UFBA. -
NLM
Brazilian Symposium on Medicinal Chemistry - BrazMedChem, 11. 2023 ;[citado 2024 out. 02 ] -
Vancouver
Brazilian Symposium on Medicinal Chemistry - BrazMedChem, 11. 2023 ;[citado 2024 out. 02 ] - Optimization of new dihydrofolate reductase inhibitors of mycobacterium tuberculosis (mtDHFR): molecular docking, synthesis, evaluation of enzyme inhibition and antimycobacterial activity
- Design, synthesis and biological activity of novel substituted 3-benzoic acid derivatives as MtDHFR inhibitors
- Using a fragment-based approach to identify alternative chemical scaffolds targeting dihydrofolate reductase from Mycobacterium tuberculosis
- Virtual screening applied in hit identification as LSD1 inhibitors, a epigenetic target for cancer treatment
- Target sites for the design of anti-trypanosomatid drugs based on the structure of dihydroorotate dehydrogenase
- QSAR studies on the human sirtuin 2 inhibition by non-covalent 7,5,2-anilinobenzamide derivatives
- Construction and validation of the 3D-structure of T. Cruzi sirtuin-2 by modeling threading
- Synthesis of two 'heteroaromatic rings of the future' for applications in medicinal chemistry
- Synthesis and docking study for compounds analogs of LSD1 inhibitor
- Insights into newly approved drugs from a medicinal chemistry perspective
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