2,2,2-Trifluoroethylamine as a peptidic bond bioisostere in reversible covalent inhibitors of cysteine proteases (2019)
- Authors:
- USP affiliated authors: MONTANARI, CARLOS ALBERTO - IQSC ; LAMEIRO, RAFAEL DA FONSECA - IQSC ; SHAMIM, ANWAR - IQSC
- Unidade: IQSC
- Subjects: SÍNTESE ORGÂNICA; DOENÇAS PARASITÁRIAS; PEPTÍDEOS
- Keywords: Bioisosteric replacement; Cysteine protease; 2,2,2-Trifluoroethylamine
- Agências de fomento:
- Language: Inglês
- Imprenta:
- Publisher: Instituto de Química de São Carlos, IQSC, Universidade de São Paulo, USP
- Publisher place: São Paulo
- Date published: 2019
- Source:
- Título do periódico: Book of Abstracts
- Conference titles: The São Carlos Special Medicinal Chemistry Meeting - SancaMedChem2019
-
ABNT
LAMEIRO, Rafael da Fonseca e SHAMIM, Anwar e MONTANARI, Carlos Alberto. 2,2,2-Trifluoroethylamine as a peptidic bond bioisostere in reversible covalent inhibitors of cysteine proteases. 2019, Anais.. São Paulo: Instituto de Química de São Carlos, IQSC, Universidade de São Paulo, USP, 2019. Disponível em: http://sancamedchem.iqsc.usp.br/files/2019/11/Book-of-abstracts-SancaMedChem2019.pdf. Acesso em: 24 abr. 2024. -
APA
Lameiro, R. da F., Shamim, A., & Montanari, C. A. (2019). 2,2,2-Trifluoroethylamine as a peptidic bond bioisostere in reversible covalent inhibitors of cysteine proteases. In Book of Abstracts. São Paulo: Instituto de Química de São Carlos, IQSC, Universidade de São Paulo, USP. Recuperado de http://sancamedchem.iqsc.usp.br/files/2019/11/Book-of-abstracts-SancaMedChem2019.pdf -
NLM
Lameiro R da F, Shamim A, Montanari CA. 2,2,2-Trifluoroethylamine as a peptidic bond bioisostere in reversible covalent inhibitors of cysteine proteases [Internet]. Book of Abstracts. 2019 ;[citado 2024 abr. 24 ] Available from: http://sancamedchem.iqsc.usp.br/files/2019/11/Book-of-abstracts-SancaMedChem2019.pdf -
Vancouver
Lameiro R da F, Shamim A, Montanari CA. 2,2,2-Trifluoroethylamine as a peptidic bond bioisostere in reversible covalent inhibitors of cysteine proteases [Internet]. Book of Abstracts. 2019 ;[citado 2024 abr. 24 ] Available from: http://sancamedchem.iqsc.usp.br/files/2019/11/Book-of-abstracts-SancaMedChem2019.pdf - Investigating the lack of translation from cruzain inhibition to Trypanosoma cruzi activity with machine learning and chemical space analyses
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