Structural basis for selective inhibition of trypanosomatid glyceraldehyde-3-phosphate dehydrogenase: molecular docking and 3D QSAR studies (2008)
- Authors:
- USP affiliated authors: OLIVA, GLAUCIUS - IFSC ; MONTANARI, CARLOS ALBERTO - IQSC ; ANDRICOPULO, ADRIANO DEFINI - IFSC
- Unidades: IFSC; IQSC
- Subjects: PLANEJAMENTO DE FÁRMACOS; TRYPANOSOMA CRUZI; LEISHMANIA; DOENÇAS PARASITÁRIAS
- Language: Inglês
- Imprenta:
- Publisher place: Washington, DC
- Date published: 2008
- Source:
- Título: Journal of Chemical Information and Modeling
- ISSN: 1549-9596
- Volume/Número/Paginação/Ano: v. 48, n. 4, p. 918-929, Apr. 2008
-
ABNT
GUIDO, Rafael Victorio Carvalho et al. Structural basis for selective inhibition of trypanosomatid glyceraldehyde-3-phosphate dehydrogenase: molecular docking and 3D QSAR studies. Journal of Chemical Information and Modeling, v. 48, n. 4, p. 918-929, 2008Tradução . . Disponível em: https://repositorio.usp.br/directbitstream/3824a029-d3d7-4653-a44d-3ebcc97b2e63/PROD014713_1666469.pdf. Acesso em: 06 maio 2026. -
APA
Guido, R. V. C., Oliva, G., Montanari, C. A., & Andricopulo, A. D. (2008). Structural basis for selective inhibition of trypanosomatid glyceraldehyde-3-phosphate dehydrogenase: molecular docking and 3D QSAR studies. Journal of Chemical Information and Modeling, 48( 4), 918-929. Recuperado de https://repositorio.usp.br/directbitstream/3824a029-d3d7-4653-a44d-3ebcc97b2e63/PROD014713_1666469.pdf -
NLM
Guido RVC, Oliva G, Montanari CA, Andricopulo AD. Structural basis for selective inhibition of trypanosomatid glyceraldehyde-3-phosphate dehydrogenase: molecular docking and 3D QSAR studies [Internet]. Journal of Chemical Information and Modeling. 2008 ; 48( 4): 918-929.[citado 2026 maio 06 ] Available from: https://repositorio.usp.br/directbitstream/3824a029-d3d7-4653-a44d-3ebcc97b2e63/PROD014713_1666469.pdf -
Vancouver
Guido RVC, Oliva G, Montanari CA, Andricopulo AD. Structural basis for selective inhibition of trypanosomatid glyceraldehyde-3-phosphate dehydrogenase: molecular docking and 3D QSAR studies [Internet]. Journal of Chemical Information and Modeling. 2008 ; 48( 4): 918-929.[citado 2026 maio 06 ] Available from: https://repositorio.usp.br/directbitstream/3824a029-d3d7-4653-a44d-3ebcc97b2e63/PROD014713_1666469.pdf - Brazilian Symposium on Medicinal Chemistry
- Avaliação do mecanismo de inibição não-específica na descoberta de inibidores enzimáticos a partir de produtos naturais
- Effects of organic solvents on the enzyme activity of Trypanosoma cruzi glyceraldehyde-3-phosphate dehydrogenase in calorimetric assays
- Discovery of novel Trypanosoma cruzi glyceraldehyde-3-phosphate dehydrogenase inhibitors
- Modelagem in silico de ADME: holograma QSAR na geração de um modelo preditivo para a ligação às proteínas plasmáticas
- Non-selective inhibition of Tryponosoma cruzi GAPDH and rabbit GAPDH determined by isothermal titration calorimetry
- Discovering novel inhibitors of Trypanosoma cruzi GAPGH: a virtual screening, calorimetric and cell assays
- Estudos de QSAR 3D e modelagem molecular de hidroxipironas como inibidores da protease do vírus HIV-1
- In silico screening for the identification of new hits of trypanosoma cruzi GAPDH
- Emprego do método volsurf na criação de um modelo preditivo de biodisponibilidade oral
Download do texto completo
| Tipo | Nome | Link | |
|---|---|---|---|
| PROD014713_1666469.pdf |
How to cite
A citação é gerada automaticamente e pode não estar totalmente de acordo com as normas
